AR227201A1 - Procedimiento para preparar polvo capaz de ser reconstituido mediante el agregado de agua para dar una suspension farmaceuticamente microcapsulas de sal de adicion de acido de bacampicilina en un medio de suspension acuosa - Google Patents
Procedimiento para preparar polvo capaz de ser reconstituido mediante el agregado de agua para dar una suspension farmaceuticamente microcapsulas de sal de adicion de acido de bacampicilina en un medio de suspension acuosaInfo
- Publication number
- AR227201A1 AR227201A1 AR286473A AR28647381A AR227201A1 AR 227201 A1 AR227201 A1 AR 227201A1 AR 286473 A AR286473 A AR 286473A AR 28647381 A AR28647381 A AR 28647381A AR 227201 A1 AR227201 A1 AR 227201A1
- Authority
- AR
- Argentina
- Prior art keywords
- water
- suspension
- reconstituted
- pharmaceutically
- give
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 239000007900 aqueous suspension Substances 0.000 title 1
- PFOLLRNADZZWEX-FFGRCDKISA-N bacampicillin Chemical compound C1([C@@H](N)C(=O)N[C@H]2[C@@H]3N(C2=O)[C@H](C(S3)(C)C)C(=O)OC(C)OC(=O)OCC)=CC=CC=C1 PFOLLRNADZZWEX-FFGRCDKISA-N 0.000 title 1
- 229960002699 bacampicillin Drugs 0.000 title 1
- 239000003094 microcapsule Substances 0.000 title 1
- 239000000843 powder Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- 239000000725 suspension Substances 0.000 title 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/180,537 US4321253A (en) | 1980-08-22 | 1980-08-22 | Suspension of microencapsulated bacampicillin acid addition salt for oral, especially pediatric, administration |
Publications (1)
Publication Number | Publication Date |
---|---|
AR227201A1 true AR227201A1 (es) | 1982-09-30 |
Family
ID=22660812
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR286473A AR227201A1 (es) | 1980-08-22 | 1981-08-19 | Procedimiento para preparar polvo capaz de ser reconstituido mediante el agregado de agua para dar una suspension farmaceuticamente microcapsulas de sal de adicion de acido de bacampicilina en un medio de suspension acuosa |
Country Status (41)
Country | Link |
---|---|
US (1) | US4321253A (en]) |
JP (1) | JPS5775986A (en]) |
KR (1) | KR860000513B1 (en]) |
AR (1) | AR227201A1 (en]) |
AT (1) | AT370994B (en]) |
AU (1) | AU529965B2 (en]) |
BE (1) | BE890028A (en]) |
BG (1) | BG42000A3 (en]) |
CA (1) | CA1137414A (en]) |
CH (1) | CH650674A5 (en]) |
CS (1) | CS225845B2 (en]) |
DD (1) | DD201644A5 (en]) |
DE (1) | DE3132614C2 (en]) |
DK (1) | DK158971C (en]) |
DZ (1) | DZ315A1 (en]) |
ES (1) | ES504905A0 (en]) |
FI (1) | FI72647C (en]) |
FR (1) | FR2488798A1 (en]) |
GB (1) | GB2082539B (en]) |
GR (1) | GR74983B (en]) |
HK (1) | HK43786A (en]) |
HU (1) | HU188679B (en]) |
IE (1) | IE51506B1 (en]) |
IL (1) | IL63617A (en]) |
IN (1) | IN156538B (en]) |
IT (1) | IT1138161B (en]) |
KE (1) | KE3626A (en]) |
LU (1) | LU83572A1 (en]) |
MX (1) | MX5731A (en]) |
MY (1) | MY8600597A (en]) |
NL (1) | NL191978C (en]) |
NO (1) | NO154821C (en]) |
NZ (1) | NZ198106A (en]) |
PH (1) | PH17125A (en]) |
PL (1) | PL232141A1 (en]) |
PT (1) | PT73555B (en]) |
RO (1) | RO82679B (en]) |
SE (1) | SE448819B (en]) |
SU (1) | SU1364226A3 (en]) |
YU (1) | YU43985B (en]) |
ZA (1) | ZA815793B (en]) |
Families Citing this family (43)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH647676A5 (fr) * | 1978-12-22 | 1985-02-15 | Donald E Panoz | Formes galeniques a usage oral, a liberation programmee et leurs procedes de preparation. |
SE8103843L (sv) * | 1981-06-18 | 1982-12-19 | Astra Laekemedel Ab | Farmaceutisk mixtur |
SE8203953D0 (sv) * | 1982-06-24 | 1982-06-24 | Astra Laekemedel Ab | Pharmaceutical mixture |
US4994260A (en) * | 1982-05-28 | 1991-02-19 | Astra Lakemedel Aktiebolag | Pharmaceutical mixture |
EP0111560A4 (en) * | 1982-06-14 | 1987-02-03 | Key Pharma | ASPIRINE WITH CONTINUOUS LEVEL. |
US4508702A (en) * | 1982-06-14 | 1985-04-02 | Key Pharmaceuticals, Inc. | Sustained release aspirin |
DE3382392D1 (de) * | 1982-07-09 | 1991-10-02 | Key Pharma | Dosierungsart zur dauerhaften verabreichung von chinidin. |
US4634587A (en) * | 1982-07-09 | 1987-01-06 | Key Pharmaceuticals, Inc. | Sustained release quinidine dosage form |
AU569277B2 (en) * | 1983-03-03 | 1988-01-28 | Dow Chemical Company, The | Aqueuos dispersion of water-insoluble organophilic cellulose ether for sustained release of active agents |
US4555399A (en) * | 1983-11-18 | 1985-11-26 | Key Pharmaceuticals, Inc. | Aspirin tablet |
IE58110B1 (en) * | 1984-10-30 | 1993-07-14 | Elan Corp Plc | Controlled release powder and process for its preparation |
SE8405611D0 (sv) * | 1984-11-09 | 1984-11-09 | Astra Laekemedel Ab | Process for stabilization of bacampicillin hydrochloride |
US4800087A (en) * | 1986-11-24 | 1989-01-24 | Mehta Atul M | Taste-masked pharmaceutical compositions |
GB8628359D0 (en) * | 1986-11-27 | 1986-12-31 | Zyma Sa | Galenical formulation |
US4853229A (en) * | 1987-10-26 | 1989-08-01 | Alza Corporation | Method for adminstering tiny pills |
US5084278A (en) * | 1989-06-02 | 1992-01-28 | Nortec Development Associates, Inc. | Taste-masked pharmaceutical compositions |
RU2123863C1 (ru) * | 1992-04-30 | 1998-12-27 | Шеринг Корпорейшн | Содержащая гидратированный цефтибутен порошковая антибактериальная композиция, предназначенная для орального использования в виде суспензии |
US6270795B1 (en) | 1995-11-09 | 2001-08-07 | Microbiological Research Authority | Method of making microencapsulated DNA for vaccination and gene therapy |
US6270804B1 (en) * | 1998-04-03 | 2001-08-07 | Biovail Technologies Ltd. | Sachet formulations |
IN191482B (en]) * | 1999-03-19 | 2003-12-06 | Ranbaxy Lab Ltd | |
JP4711478B2 (ja) * | 1999-08-13 | 2011-06-29 | 旭化成ケミカルズ株式会社 | 味がマスクされた薬物 |
US20050037086A1 (en) * | 1999-11-19 | 2005-02-17 | Zycos Inc., A Delaware Corporation | Continuous-flow method for preparing microparticles |
SK8562002A3 (en) | 1999-12-23 | 2003-10-07 | Pfizer Prod Inc | Pharmaceutical compositions providing enhanced drug concentrations |
EP1118333A1 (en) * | 2000-01-18 | 2001-07-25 | Eurand International S.P.A. | Compositions with enhanced oral bioavailability |
DE60128215T2 (de) | 2000-04-20 | 2008-01-10 | Novartis Ag | Beschichtungszusammensetzung zur geschmacksmaskierung |
US6551617B1 (en) | 2000-04-20 | 2003-04-22 | Bristol-Myers Squibb Company | Taste masking coating composition |
EP1292285A4 (en) * | 2000-06-02 | 2009-07-22 | Eisai Corp North America | SYSTEMS FOR DISPENSING BIOACTIVE AGENTS |
FR2822834B1 (fr) * | 2001-04-02 | 2005-02-25 | Flamel Tech Sa | Suspension colloidale de nanoparticules a base de copolymeres amphiphile pour la vectorisation de principes actifs et leur mode de preparation |
CA2447693A1 (en) * | 2001-05-31 | 2002-12-05 | Cima Labs Inc. | Taste-masking of highly water-soluble drugs |
KR20030015655A (ko) * | 2001-08-17 | 2003-02-25 | 한미약품공업 주식회사 | 항암제의 경구흡수율을 증가시키는 인단계 화합물의결정성 산부가염, 이의 제조방법 및 이를 함유하는 약학적조성물 |
FR2830447B1 (fr) * | 2001-10-09 | 2004-04-16 | Flamel Tech Sa | Forme galenique orale microparticulaire pour la liberation retardee et controlee de principes actifs pharmaceutiques |
US8101209B2 (en) * | 2001-10-09 | 2012-01-24 | Flamel Technologies | Microparticulate oral galenical form for the delayed and controlled release of pharmaceutical active principles |
CA2480826C (fr) | 2002-04-09 | 2012-02-07 | Flamel Technologies | Formulation pharmaceutique orale sous forme de suspension aqueuse de microcapsules permettant la liberation modifiee de principe(s) actif(s) |
KR20050005437A (ko) * | 2002-04-09 | 2005-01-13 | 플라멜 테크놀로지스 | 아목시실린의 변형 방출을 위한 마이크로캡슐 수성 현탁액형태의 경구 제약학적 제제 |
FR2842736B1 (fr) | 2002-07-26 | 2005-07-22 | Flamel Tech Sa | Formulation pharmaceutique orale sous forme d'une pluralite de microcapsules permettant la liberation prolongee de principe(s) actif(s) peu soluble(s) |
FR2842735B1 (fr) * | 2002-07-26 | 2006-01-06 | Flamel Tech Sa | Microcapsules a liberation modifiee de principes actifs peu solubles pour l'administration per os |
FR2843117B1 (fr) * | 2002-07-30 | 2004-10-15 | Flamel Tech Sa | Polyaminoacides fonctionnalises par au moins un groupement hydrophobe et leurs applications notamment therapeutiques |
US7632521B2 (en) * | 2003-07-15 | 2009-12-15 | Eurand, Inc. | Controlled release potassium chloride tablets |
FR2860516B1 (fr) * | 2003-10-03 | 2006-01-13 | Flamel Tech Sa | Homopolyaminoacides telecheliques fonctionnalises par des groupements hydrophobes et leurs applications notamment therapeutiques |
FR2862536B1 (fr) * | 2003-11-21 | 2007-11-23 | Flamel Tech Sa | Formulations pharmaceutiques pour la liberation prolongee de principe(s) actif(s), ainsi que leurs applications notamment therapeutiques |
US7244765B2 (en) * | 2004-06-25 | 2007-07-17 | Cytokine Pharmasciences, Inc | Guanylhydrazone salts, compositions, processes of making and methods of using |
FR2885526B1 (fr) * | 2005-05-13 | 2007-07-27 | Flamel Technologies Sa | Medicament oral a base d'inhibiteur de pompe a protons |
US20180177820A1 (en) * | 2015-10-13 | 2018-06-28 | Techno Guard Co. Ltd. | Protective composition for gastrointestinal mucosa |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3549746A (en) * | 1967-11-02 | 1970-12-22 | Bristol Myers Co | Antibiotic composition |
US3873521A (en) * | 1970-09-17 | 1975-03-25 | Astra Laekemedel Ab | Esters of {60 -amino penicillins |
ZA718014B (en) | 1970-12-23 | 1972-08-30 | Beecham Group Ltd | Pharmaceutical formulations |
US4016254A (en) * | 1972-05-19 | 1977-04-05 | Beecham Group Limited | Pharmaceutical formulations |
GB1455296A (en) * | 1973-05-24 | 1976-11-10 | Beecham Group Ltd | Veterinary treatment |
GB1479655A (en) | 1974-03-08 | 1977-07-13 | Beecham Group Ltd | Antibiotic preparations |
US4127647A (en) * | 1975-04-08 | 1978-11-28 | Meiji Seika Kaisha, Ltd. | Process for preparation of stable amorphous macrolide antibiotic solids |
JPS5840529B2 (ja) * | 1975-09-29 | 1983-09-06 | 明治製菓株式会社 | ケイコウヨウセイザイノセイホウ |
GB1561301A (en) * | 1976-01-02 | 1980-02-20 | Beecham Group Ltd | Orally administrable pharmaceutical composition |
ZA793934B (en) * | 1978-08-04 | 1980-07-30 | Beecham Group Ltd | Powders |
JPS57105316A (en) * | 1980-12-23 | 1982-06-30 | Hitachi Cable Ltd | Method of fitting heat-shrinkable tube |
-
1980
- 1980-08-22 US US06/180,537 patent/US4321253A/en not_active Expired - Lifetime
-
1981
- 1981-06-23 IN IN405/DEL/81A patent/IN156538B/en unknown
- 1981-07-08 RO RO104817A patent/RO82679B/ro unknown
- 1981-07-08 DZ DZ816254A patent/DZ315A1/fr active
- 1981-07-09 HU HU812005A patent/HU188679B/hu unknown
- 1981-07-09 SU SU813310057A patent/SU1364226A3/ru active
- 1981-07-10 CS CS815334A patent/CS225845B2/cs unknown
- 1981-07-10 PL PL23214181A patent/PL232141A1/xx unknown
- 1981-07-10 BG BG052867A patent/BG42000A3/xx unknown
- 1981-08-05 GB GB8123977A patent/GB2082539B/en not_active Expired
- 1981-08-14 CH CH5277/81A patent/CH650674A5/fr not_active IP Right Cessation
- 1981-08-18 DE DE3132614A patent/DE3132614C2/de not_active Expired
- 1981-08-19 AT AT0362781A patent/AT370994B/de not_active IP Right Cessation
- 1981-08-19 GR GR65819A patent/GR74983B/el unknown
- 1981-08-19 AR AR286473A patent/AR227201A1/es active
- 1981-08-19 CA CA000384168A patent/CA1137414A/en not_active Expired
- 1981-08-20 BE BE0/205725A patent/BE890028A/fr not_active IP Right Cessation
- 1981-08-20 PH PH26070A patent/PH17125A/en unknown
- 1981-08-20 IT IT23587/81A patent/IT1138161B/it active
- 1981-08-20 YU YU2017/81A patent/YU43985B/xx unknown
- 1981-08-20 IE IE1911/81A patent/IE51506B1/en not_active IP Right Cessation
- 1981-08-20 DD DD81232705A patent/DD201644A5/de not_active IP Right Cessation
- 1981-08-20 FI FI812574A patent/FI72647C/fi not_active IP Right Cessation
- 1981-08-20 NZ NZ198106A patent/NZ198106A/xx unknown
- 1981-08-20 IL IL63617A patent/IL63617A/xx not_active IP Right Cessation
- 1981-08-20 LU LU83572A patent/LU83572A1/fr unknown
- 1981-08-21 FR FR8116074A patent/FR2488798A1/fr active Granted
- 1981-08-21 ES ES504905A patent/ES504905A0/es active Granted
- 1981-08-21 NO NO812827A patent/NO154821C/no unknown
- 1981-08-21 SE SE8104974A patent/SE448819B/sv not_active IP Right Cessation
- 1981-08-21 NL NL8103902A patent/NL191978C/xx not_active IP Right Cessation
- 1981-08-21 DK DK372181A patent/DK158971C/da not_active IP Right Cessation
- 1981-08-21 PT PT73555A patent/PT73555B/pt unknown
- 1981-08-21 AU AU74416/81A patent/AU529965B2/en not_active Expired
- 1981-08-21 ZA ZA815793A patent/ZA815793B/xx unknown
- 1981-08-21 JP JP56131418A patent/JPS5775986A/ja active Granted
- 1981-08-21 KR KR1019810003057A patent/KR860000513B1/ko not_active Expired
- 1981-08-24 MX MX573181A patent/MX5731A/es unknown
-
1986
- 1986-04-04 KE KE3626A patent/KE3626A/xx unknown
- 1986-06-09 HK HK437/86A patent/HK43786A/xx not_active IP Right Cessation
- 1986-12-30 MY MY597/86A patent/MY8600597A/xx unknown
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